Pharmacologie

9 décembre 2024

Diversity-oriented synthesis of second generation guanidinium-rich transporters toward cell-selective penetration

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Auteurs et autrices

Duc Tai Nguyen, Michael Desgagné, Andréanne Laniel, Christine Lavoie, Pierre-Luc Boudreault

14 novembre 2024

Discovery and Preclinical Characterization of Fulacimstat (BAY 1142524), a Potent and Selective Chymase Inhibitor As a New Profibrinolytic Approach for Safe Thrombus Resolution

Auteurs et autrices

Chantal Fürstner, Jens Ackerstaff, Heinrich Meier, Alexander Straub, Joachim Mittendorf, Jens Schamberger, Martina Schäfer, Kirsten Börngen, Hannah Jörißen, Dmitry Zubov, Katja Zimmermann, Adrian Tersteegen, Volker Geiss, Elke Hartmann, Barbara Albrecht-Küpper, Pedro D'Orléans-Juste, Catherine Lapointe, Laurence Vincent, Stefan Heitmeier, Hanna Tinel

24 octobre 2024

Diversity-oriented synthesis of second generation guanidinium-rich transporters toward cell-selective penetration

Discovery and Preclinical Characterization of Fulacimstat (BAY 1142524), a Potent and Selective Chymase Inhibitor As a New Profibrinolytic Approach for Safe Thrombus Resolution

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